GW791343 | P2X7 antagonist | Probechem Biochemicals

Chemical Structure : GW791343

GW791343 (GW791343 dihydrochloride)

Catalog No.: PC-25894Not For Human Use, Lab Use Only.

GW791343 dihydrochloride is a selective, allosteric antagonist with negative allosteric effects at the human P2X7 receptor with pIC50 of 6.9-7.2, but is a positive allosteric modulator of the rat P2X(7) receptor.

Packing	Price	Stock	Quantity
50 mg		Get quote
100 mg		Get quote
250 mg		Get quote

Get Quotation Now

* Please select Quantity before adding items.

or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Biological Activity

Physicochemical Properties

M.Wt	447.35
Formula	C20H26Cl2F2N4O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-((3,4-Difluorophenyl)amino)-N-(2-methyl-5-(piperazin-1-ylmethyl)phenyl)acetamide dihydrochloride

References

1. Michel AD, et al. Br J Pharmacol. 2008 Feb;153(4):737-50.

2. Michel AD, et al. Br J Pharmacol. 2008 Nov;155(5):738-51.

Overnight Delivery
Fast & Safe Delivery Worldwide
Rewards Program

About Us

Our Services

Site Map

Join with Us
Product Use Citations

Pharmacological Glossary Abbreviations

Abbreviations

Quality Manual

Inquiry Form
How to Order

Terms & Conditions

Credit Card Payment

Shipping Rates & Policies

Privacy Policy
sales@probechem.com

GW791343 (GW791343 dihydrochloride)

Biological Activity

Physicochemical Properties

References

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

Get Quote

* Indicates a Required FieldYour information is safe with us.