Chemical Structure : GeA-69
Catalog No.: PC-60021Not For Human Use, Lab Use Only.
GeA-69 (GeA69) is a potent, selective, allosteric, cell-active PARP14 macrodomain 2 (MD2) inhibitor with Kd of 0.86 uM in ITC assays.
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GeA-69 (GeA69) is a potent, selective, allosteric, cell-active PARP14 macrodomain 2 (MD2) inhibitor with Kd of 0.86 uM in ITC assays; displays high selectivity over other human macrodomains; engages PARP14 MD2 in intact cells and prevents its localization to sites of DNA damage.
M.Wt | 300.361 | |
Formula | C20H16N2O | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
1. Schuller M, et al. ACS Chem Biol. 2017 Nov 17;12(11):2866-2874.
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