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Chemical Structure : KDM5-C49
CAS No.: 1596348-16-1
Catalog No.: PC-62294Not For Human Use, Lab Use Only.
KDM5-C49 is a potent, selective KDM5 inhibitor with IC50 of 25, 30 and 59 nM for KDM5A, B and C, respectively.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $248 | In stock | |
| 10 mg | $398 | In stock | |
| 25 mg | $598 | In stock | |
| 100 mg | Get quote |
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KDM5-C49 is a potent, selective KDM5 inhibitor with IC50 of 25, 30 and 59 nM for KDM5A, B and C, respectively.
KDM5-C49 displays 25-100-fold selectivity over KDM6B, 2-30-fold selectivity over KDM4 family, but with less cell-permeablity.
| M.Wt | 308.382 | |
| Formula | C15H24N4O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
2-(((2-((2-(dimethylamino)ethyl)(ethyl)amino)-2-oxoethyl)amino)methyl)isonicotinic acid |
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1. Johansson C, et. Nat Chem Biol. 2016 Jul;12(7):539-45.
2. Horton JR, et al. Cell Chem Biol. 2016 Jul 21;23(7):769-81.
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