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Chemical Structure : LDN-27219
CAS No.: 312946-37-5
Catalog No.: PC-45039Not For Human Use, Lab Use Only.
LDN-27219 is a potent, reversible inhibitor of hTGase (Tissue transglutaminase) with IC50 of 0.8 uM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $98 | In stock | |
| 25 mg | $158 | In stock | |
| 50 mg | $258 | In stock | |
| 100 mg | Get quote |
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LDN-27219 is a potent, reversible inhibitor of hTGase (Tissue transglutaminase) with IC50 of 0.8 uM.
LDN-27219 does not bind at the enzyme's active site but rather at the enzyme's GTP site, or a site that regulates binding of GTP.
| M.Wt | 408.4966 | |
| Formula | C20H16N4O2S2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: ≥ 4.3 mg/mL |
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| Chemical Name/SMILES |
Acetic acid, 2-[(3,4-dihydro-4-oxo-3,5-diphenylthieno[2,3-d]pyrimidin-2-yl)thio]-, hydrazide |
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1. Duval E, et al. Bioorg Med Chem Lett. 2005 Apr 1;15(7):1885-9.
2. Case A, et al. Biochemistry. 2007 Jan 30;46(4):1106-15.
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