LP-360924 | GPR139 agonist | Probechem Biochemicals

Chemical Structure : LP-360924

LP-360924 (LP360924)

Catalog No.: PC-26123Not For Human Use, Lab Use Only.

LP-360924 is a potent, selective GPR139 agonist, stimulates cAMP production in cAMP assays.

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Biological Activity

LP-360924 is a potent, selective GPR139 agonist, stimulates cAMP production in cAMP assays.
LP-360924 stimulation increased cAMP production by 8- to 10-fold in GPR139 cells, does not show any activity in β2 AR cells at concentrations up to 100 uM.
LP-360924 stimulated cAMP production only in GPR139-transfected cells, not in vector or β2 AR-transfected cells.

Physicochemical Properties

M.Wt	562.65
Formula	C26H30N10O3S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(2-((4-methoxy-6-((3-methoxypropyl)amino)-1,3,5-triazin-2-yl)amino)-4-phenylthiazol-5-yl)(4-(pyrimidin-2-yl)piperazin-1-yl)methanone

References

1. Hu LA, et al. J Biomol Screen. 2009 Aug;14(7):789-97.

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LP-360924 (LP360924)

Biological Activity

Physicochemical Properties

References

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