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Lorundrostat

Chemical Structure : Lorundrostat

CAS No.: 1820940-17-7

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Lorundrostat (MT-4129, MT4129)

Catalog No.: PC-24474Not For Human Use, Lab Use Only.

Lorundrostat (MT-4129) is a highly selective inhibitor of CYP11B2 (aldosterone synthase) Ki values of 1.27 nM for hCYP11B2 and 475 nM for hCYP11B1, reduces systolic blood pressure.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Lorundrostat (MT-4129) is a highly selective inhibitor of CYP11B2 (aldosterone synthase) Ki values of 1.27 nM for hCYP11B2 and 475 nM for hCYP11B1, reduces systolic blood pressure.

Physicochemical Properties

M.Wt 451.58
Formula C24H33N7O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

N-(trans-4-Acetamidocyclohexyl)-2-(4-(5-(p-tolyl)-1,2,4-triazin-3-yl)piperazin-1-yl)acetamide

References

1. Laffin LJ, et al. JAMA. 2023 Sep 26;330(12):1140-1150.

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