M085 | TRPC3/6/7 activator | Probechem Biochemicals

Chemical Structure : M085

Catalog No.: PC-21344Not For Human Use, Lab Use Only.

M085 (TRPC3/6/7 activator 4o) is a potent and selective TRPC3/6/7 activator with EC50 of 4.66 uM, also activates hTRPC6 with EC50 of 3.8 uM.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

M085 (TRPC3/6/7 activator 4o) is a potent and selective TRPC3/6/7 activator with EC50 of 4.66 uM, also activates hTRPC6 with EC50 of 3.8 uM.

M.Wt	398.44
Formula	C21H23FN4O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4-(3-(4-fluorophenyl)-7-hydroxy-2-methylpyrazolo[1,5-a]pyrimidin-5-yl)piperidin-1-yl propionate

1. Qu C., et al. J. Med. Chem. 2017;60:4680–4692.

2. Yang PL, et al. J Biol Chem. 2021 Oct;297(4):101125.