You are here:Home-Chemical Inhibitors & Agonists-Metabolic Enzyme/Protease-Pyruvate Dehydrogenase Kinase (PDK)-M77976
M77976

Chemical Structure : M77976

CAS No.: 394237-61-7

M77976 (M 77976)

Catalog No.: PC-21872Not For Human Use, Lab Use Only.

M77976 is a selective inhibitor of pyruvate dehydrogenase kinase 4 (PDK4) with IC50 of 648 uM, binds to the ATP-binding pocket of PDK4.

Packing Price Stock Quantity
5 mg $148 In stock
10 mg $238 In stock
25 mg $358 In stock
50 mg Get quote
100 mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

M77976 is a selective inhibitor of pyruvate dehydrogenase kinase 4 (PDK4) with IC50 of 648 uM, binds to the ATP-binding pocket of PDK4.

Physicochemical Properties

M.Wt 296.33
Formula C17H16N2O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

4-(4-(4-methoxyphenyl)-5-methyl-1H-pyrazol-3-yl)benzene-1,3-diol

References

1. Kukimoto-Niino M, et al. Acta Crystallogr D Biol Crystallogr. 2011 Sep;67(Pt 9):763-73.

2. Wang H, et al. Cancer Metab. 2024 Jan 10;12(1):2.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: