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Chemical Structure : MCL0020
CAS No.: 475498-26-1
Catalog No.: PC-21480Not For Human Use, Lab Use Only.
MCL0020 is a potent, selective inverse agonist of melanocortin MC4 receptor (MC4R) with binding IC50 of 11.6 nM, shows negligible affinity for MC1 and MC3 receptors.
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MCL0020 is a potent, selective inverse agonist of melanocortin MC4 receptor (MC4R) with binding IC50 of 11.6 nM, shows negligible affinity for MC1 and MC3 receptors.
MCL0020 attenuates swim stress-induced anxiogeniclike behavior in light/dark exploration tests in mice, significantly reverses stress-induced anorexia in rats.
| M.Wt | 609.72 | |
| Formula | C34H39N7O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
N-Acetyl-3-(2-naphthalenyl)-D-alanyl-L-arginyl-3-(2-naphthalenyl)-L-alaninamide |
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1. Chaki S, et al. Eur J Pharmacol. 2003 Aug 1;474(1):95-101.
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