Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.

You are here:Home-Chemical Inhibitors & Agonists-GPCR-Cannabinoid Receptor-MDA77
MDA77

Chemical Structure : MDA77

CAS No.: 1103774-21-5

MDA77

Catalog No.: PC-26031Not For Human Use, Lab Use Only.

MDA77 is a potent selective cannabinoid receptor 2 (CB2) inverse agonist with EC50 of 5.82 nM at human CB2, with no activity at CB1, inhibits the effect of MDA7 (CB2 agonist) in animal model of neuropathic pain.

Packing Price Stock Quantity
50 mg Get quote
100 mg Get quote
250 mg Get quote

Bulk size, bulk discount!

Welcome credit card payment!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC)

Biological Activity

MDA77 is a potent selective cannabinoid receptor 2 (CB2) inverse agonist with EC50 of 5.82 nM at human CB2, with no activity at CB1, inhibits the effect of MDA7 (CB2 agonist) in animal model of neuropathic pain.

Physicochemical Properties

M.Wt 365.43
Formula C21H23N3O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

Benzoic acid, (2Z)-2-(1,2-dihydro-6-methoxy-2-oxo-1-pentyl-3H-indol-3-ylidene)hydrazide

References

1. Philippe Diaz, et al. J Med Chem. 2009 Jan 22;52(2):433-44.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: