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Chemical Structure : MPC-3100
Catalog No.: PC-60471Not For Human Use, Lab Use Only.
MPC-3100 is a novel potent, selective, orally bioavailable Hsp90 inhibitor with IC50 of 0.14 uM.
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MPC-3100 is a novel potent, selective, orally bioavailable Hsp90 inhibitor with IC50 of 0.14 uM.
MPC-3100 displays antiproliferative activity against a panel of cancer cell lines with IC50 of <1 uM.
MPC-3100 exhibits good in vitro profiles and a characteristic molecular biomarker signature of Hsp90 inhibition both in vitro and in vivo, shows significant antitumor effects in multiple human cancer xenograft models.
| M.Wt | 549.4 | |
| Formula | C22H25BrN6O4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Kim SH, et al. J Med Chem. 2012 Sep 13;55(17):7480-501.
2. Kim SH, et al. Bioorg Med Chem Lett. 2015 Nov 15;25(22):5254-7.
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