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MRS4478

Chemical Structure : MRS4478

CAS No.:

MRS4478 (MRS 4478;MRS-4478)

Catalog No.: PC-35049Not For Human Use, Lab Use Only.

MRS4478 is a potent, highly specific amtagonist of P2Y14 receptor with IC50 of 269 nM, does not display extensive off-target interactions with biogenic amine receptors..

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

MRS4478 is a potent, highly specific amtagonist of P2Y14 receptor with IC50 of 269 nM, does not display extensive off-target interactions with biogenic amine receptors.

Physicochemical Properties

M.Wt 452.393
Formula C23H15F3N4O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

4'-Carbamoyl-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol1-yl)-[1,1'-biphenyl]-3-carboxylic acid

References

1. Yu J, et al. J Med Chem. 2018 May 16. doi: 10.1021/acs.jmedchem.8b00168.

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