MRS8432

Chemical Structure : MRS8432

Catalog No.: PC-26269Not For Human Use, Lab Use Only.

MRS8432 is a specific stimulator of ABCG2 (breast cancer resistance protein, BCRP) ATPase activity with EC50 of 17.5 nM.

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Biological Activity

MRS8432 is a specific stimulator of ABCG2 (breast cancer resistance protein, BCRP) ATPase activity with EC50 of 17.5 nM.

M.Wt	694.10
Formula	C35H26ClF2N9O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(1S,2R,3S,4R,5S)-4-(6-((3-(4-(4-Chlorophenyl)-1H-1,2,3-triazol-1-yl)phenyl)amino)-2-((3,4-difluorophenyl)ethynyl)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide

1. Murakami M, et al. J Med Chem. 2026 Feb 26;69(4):4945-4968.