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Olorinab

Chemical Structure : Olorinab

CAS No.: 1268881-20-4

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Olorinab (APD371, APD-371)

Catalog No.: PC-60146Not For Human Use, Lab Use Only.

Olorinab (APD371) is a potent, selective and orally available CB2 cannabinoid receptor agonist with EC50 of 6.2 nM.

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5 mg $128 In stock
10 mg $198 In stock
25 mg $358 In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Olorinab (APD371) is a potent, selective and orally available CB2 cannabinoid receptor agonist with EC50 of 6.2 nM.
Olorinab (APD371) displays no activity against CB1 receptors (EC50>10 uM).
Olorinab (APD371) exhibits activity in rat model of osteoarthritis pain.

Physicochemical Properties

M.Wt 357.414
Formula C18H23N5O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

3-((4aS,5aS)-3-(((S)-1-hydroxy-3,3-dimethylbutan-2-yl)carbamoyl)-4,4a,5,5a-tetrahydro-1H-cyclopropa[4,5]cyclopenta[1,2-c]pyrazol-1-yl)pyrazine 1-oxide

References

1. Sangdon Han, et al. ACS Med. Chem. Lett., 2017, 8 (12), pp 1309-1313.

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