Chemical Structure : PD149163
CAS No.:
169528-11-4
PD149163
(PD-149163, PD 149163)
Catalog No.: PC-28013Not For Human Use, Lab Use Only.
PD149163 (PD-149163) is a reduced amide neurotensin(8-13) mimetic and selective, brain-penetrating neurotensin-1 receptor (NTR1, NTSR1) agonist, shows antipsychotic-like effects.
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Purity & Documentation Purity:
>98% (HPLC)
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Biological Activity
PD149163 (PD-149163) is a reduced amide neurotensin(8-13) mimetic and selective, brain-penetrating neurotensin-1 receptor (NTR1, NTSR1) agonist, shows antipsychotic-like effects.
Physicochemical Properties
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M.Wt
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798.07
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Formula
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C42H71N9O6
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Appearance
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Solid
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CAS No.
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Storage
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- Solide Powder
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-20°C 12 Months; 4°C 6 Months
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- In Solvent
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-80°C 6 Months; -20°C 6 Months
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Shipping
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Solubility
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10 mM in DMSO
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Chemical Name/SMILES
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{Lys(N2-[(2S)-2,6-diaminohexyl])}-Pro-Trp-{Tle}-{Leu(Et)}
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References
1. Feifel D, et al. J Pharmacol Exp Ther. 1999 Feb;288(2):710-3.
2. Norman C, et al. J Psychopharmacol. 2010 Mar;24(3):373-81.
3. Feifel D, et al. Neuropsychopharmacology. 2003 Apr;28(4):651-3.
4. Wustrow DJ, et al. Bioorg Med Chem Lett 5: 998-1002.
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