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Chemical Structure : PF-03716556
Catalog No.: PC-62889Not For Human Use, Lab Use Only.
PF-03716556 is a potent, selective, competitive and reversible gastric H+,K+-ATPase with pIC50 of 7.0 in porcine ion-tight membrane vesicle.
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PF-03716556 is a potent, selective, competitive and reversible gastric H+,K+-ATPase with pIC50 of 7.0 in porcine ion-tight membrane vesicle; exhibits highly selective profile including the canine kidney Na+,K+-ATPase; inhibited gastric acid secretion in heidenhain pouch dogs (0.3-3mg/kg, p.o.), shows potentiation for the treatment of gastroesophageal reflux disease; orally biovailable.
| M.Wt | 394.5 | |
| Formula | C22H26N4O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Mori H, et al. J Pharmacol Exp Ther. 2009 Feb;328(2):671-9.
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