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PF-04756956

Chemical Structure : PF-04756956

CAS No.: 1228934-52-8

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PF-04756956 (PF04756956, PF 04756956)

Catalog No.: PC-70198Not For Human Use, Lab Use Only.

PF-04756956 is a potent, selective CCK1 receptor agonist with EC50 of 0.47 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    PF-04756956 is a potent, selective CCK1 receptor agonist with EC50 of 0.47 nM.
    PF-04756956 elicits no biological response at the CCK2 receptors.
    PF-04756956 demonstrates robust weight loss in a diet-induced obese rat model with very low systemic exposure.

    Physicochemical Properties

    M.Wt 649.799
    Formula C40H39N7O2
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (4S)-4-((1H-indazol-3-yl)methyl)-6-(2-((R)-2-(3,5-dimethylbenzyl)piperidin-1-yl)-2-oxoethyl)-1-phenyl-4H-benzo[b][1,2,4]triazolo[4,3-d][1,4]diazepin-5(6H)-one

    References

    1. Desai AJ, et al. J Med Chem. 2015 Dec 24;58(24):9562-77.

    2. Cameron KO, et al. Bioorg Med Chem Lett. 2012 Apr 15;22(8):2943-7.

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