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Chemical Structure : PF-06462894
Catalog No.: PC-61058Not For Human Use, Lab Use Only.
A potent, subtype-selective mGluR5 negative allosteric modulator with Ki of 6.1 nM.
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A potent, subtype-selective mGluR5 negative allosteric modulator with Ki of 6.1 nM; possesses favorable properties and a predicted low clinical dose (2 mg twice daily), does not show any evidence of immune activation in a mouse drug allergy model.
| M.Wt | 329.4 | |
| Formula | C18H23N3O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Stepan AF, et al. J Med Chem. 2017 Sep 28;60(18):7764-7780.
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