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PF-07976016

Chemical Structure : PF-07976016

CAS No.: 3059496-70-4

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PF-07976016 (PF07976016)

Catalog No.: PC-28066Not For Human Use, Lab Use Only.

PF-07976016 is a potent, orally active glucose-dependent insulinotropic polypeptide receptor (GIPR) antagonist with IC50 of 4.1 nM, shows competitively binding to GIPR and blocking the increase in Gαs-mediated cAMP production induced by GIP agonists.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

PF-07976016 is a potent, orally active glucose-dependent insulinotropic polypeptide receptor (GIPR) antagonist with IC50 of 4.1 nM, shows competitively binding to GIPR and blocking the increase in Gαs-mediated cAMP production induced by GIP agonists.

Physicochemical Properties

M.Wt 471.56
Formula C28H29N3O4
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(R)-4'-(1-((4-Isopropylphenyl)carbamoyl)pyrrolidine-2-carboxamido)-[1,1'-biphenyl]-4-carboxylic acid

References

1. Patent WO2024214038 A1 2024-10-17.

2. Patent US20250235460 A1.

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