PG01037 dihydrochloride | D3R antagonist

Chemical Structure : PG01037 dihydrochloride

CAS No.: 675599-62-9

PG01037 dihydrochloride (PG-01037)

Catalog No.: PC-26861Not For Human Use, Lab Use Only.

PG01037 dihydrochloride is a potent selective dopamine D3 receptor (D3R) antagonist with binding Ki of 0.7 nM, displays 133- and 540-fold selectivity over D2 and D4 receptors, respectively.

Packing	Price	Stock
10 mg	$88	In stock
25 mg	$138	In stock
50 mg	$228	In stock
100 mg		Get quote

Get Quotation Now

* Please select Quantity before adding items.

or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Biological Activity

PG01037 dihydrochloride is a potent selective dopamine D3 receptor (D3R) antagonist with binding Ki of 0.7 nM, displays 133- and 540-fold selectivity over D2 and D4 receptors, respectively.

Physicochemical Properties

M.Wt	554.34
Formula	C26H28Cl4N4O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(E)-N-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)but-2-en-1-yl)-4-(pyridin-2-yl)benzamide dihydrochloride

References

1. Grundt P, et al. J Med Chem. 2007 Aug 23;50(17):4135-46.

Overnight Delivery
Fast & Safe Delivery Worldwide
Rewards Program

About Us

Our Services

Site Map

Join with Us
Product Use Citations

Pharmacological Glossary Abbreviations

Abbreviations

Quality Manual

Inquiry Form
How to Order

Terms & Conditions

Credit Card Payment

Shipping Rates & Policies

Privacy Policy
sales@probechem.com

PG01037 dihydrochloride (PG-01037)

Biological Activity

Physicochemical Properties

References

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

Get Quote

* Indicates a Required FieldYour information is safe with us.