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Chemical Structure : PI3Kδ-IN-7n
Catalog No.: PC-62806Not For Human Use, Lab Use Only.
PI3Kδ-IN-7n is a highly potent and selective PI3Kδ inhibitor with IC50 of 0.9 nM, displays high selectivity (>1,500-fold) over PI3Kα, PI3Kβ, PI3Kγ (IC50>1.5 uM).
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PI3Kδ-IN-7n is a highly potent and selective PI3Kδ inhibitor with IC50 of 0.9 nM, displays high selectivity (>1,500-fold) over PI3Kα, PI3Kβ, PI3Kγ (IC50>1.5 uM); shows reasonable pharmacokinetics with good bioavailability and moderate in vivo half-life; one of the most selective PI3Kδ inhibitors published to date.
| M.Wt | 429.459 | |
| Formula | C23H20FN7O | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Terstiege I, et al. Bioorg Med Chem Lett. 2017 Feb 1;27(3):679-687.
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