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PITCOIN2

Chemical Structure : PITCOIN2

CAS No.: 2397679-77-3

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PITCOIN2 (LU-06-006)

Catalog No.: PC-20451Not For Human Use, Lab Use Only.

PITCOIN2 (LU-06-006) is a potent selective PI3KC2α inhibitor with IC50 of 126 nM, has selectivity against PI3KC2γ but shows micromolar activity on PI3KC2β.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    PITCOIN2 (LU-06-006) is a potent selective PI3KC2α inhibitor with IC50 of 126 nM, has selectivity against PI3KC2γ but shows micromolar activity on PI3KC2β.

    Physicochemical Properties

    M.Wt 516.59
    Formula C25H20N6O3S2
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    N-(4-(3-hydroxyphenyl)thiazol-2-yl)-2-((4-oxo-3-phenethyl-3,4-dihydropteridin-2-yl)thio)acetamide

    References

    1. Lo WT, et al. Nat Chem Biol. 2023 Jan;19(1):18-27.

    2. Patent WO2019234237 A1.

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