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Chemical Structure : PRE-084 hydrochloride
CAS No.: 75136-54-8
Catalog No.: PC-45419Not For Human Use, Lab Use Only.
PRE-084 is a highly potent, selective sigma-1 receptor agonist with Ki of 2.2 nM, IC50 of 44 nM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 25 mg | $158 | In stock | |
| 50 mg | $258 | In stock | |
| 100 mg | $398 | In stock | |
| 200 mg | Get quote | ||
| 1 g | Get quote |
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PRE-084 is a highly potent, selective sigma-1 receptor agonist with Ki of 2.2 nM, IC50 of 44 nM.
PRE-084 shows little or no affinity for sigma-2 and PCP receptors (Ki>10 uM).
PRE-084 has nootropic and antidepressant actions in vivo, as well as antitussive and reinforcing effects.
| M.Wt | 353.8835 | |
| Formula | C19H28ClNO3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: ≥ 34 mg/mL |
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| Chemical Name/SMILES |
Cyclohexanecarboxylic acid, 1-phenyl-, 2-(4-morpholinyl)ethyl ester, hydrochloride (1:1) |
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1. Su TP, et al. J Pharmacol Exp Ther. 1991 Nov;259(2):543-50.
2. Brown C, et al. Br J Pharmacol. 2004 Jan;141(2):233-40.
3. Maurice T, et al. Br J Pharmacol. 2001 Dec;134(8):1731-41.
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