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PSB-1011

Chemical Structure : PSB-1011

CAS No.: 4499-01-8

PSB-1011

Catalog No.: PC-26167Not For Human Use, Lab Use Only.

PSB-1011 is a potent, moderately selective rat P2X2 receptor antagonist with IC50 of 79 nM, weakly inhibits P2X1 and P2X3 receptors and shows no activity against P2X4 and P2X7 receptors.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

PSB-1011 is a potent, moderately selective rat P2X2 receptor antagonist with IC50 of 79 nM, weakly inhibits P2X1 and P2X3 receptors and shows no activity against P2X4 and P2X7 receptors.

Physicochemical Properties

M.Wt 681.38
Formula C23H12Cl2N6Na2O8S2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

sodium 1-amino-4-((3-((4,6-dichloro-1,3,5-triazin-2-yl)amino)-4-sulfonatophenyl)amino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate

References

1. Baqi Y, et al. J Med Chem. 2011;54:817–830.

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