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Chemical Structure : PSB-16671
Catalog No.: PC-72359Not For Human Use, Lab Use Only.
PSB-16671 is a novel orthosteric and allosteric activator of GPR84, activates human GPR84 with EC50 of 41.3 nM in cAMP accumulation assays.
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PSB-16671 is a novel orthosteric and allosteric activator of GPR84, activates human GPR84 with EC50 of 41.3 nM in cAMP accumulation assays.
PSB-16671 is selective versus related fatty acid receptors and the arylhydrocarbon receptor.
PSB-16671 shows an EC50 of 5.47 uM in β-Arrestin assays, and allosteric KB value of 634 nM.
| M.Wt | 318.275 | |
| Formula | C17H10F4N2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Sarah J Mancini, et al. Sci Rep. 2019 Feb 12;9(1):1861.
2. Pillaiyar T, et al. J Med Chem. 2017 May 11;60(9):3636-3655.
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