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Chemical Structure : RLX-33
Catalog No.: PC-38726Not For Human Use, Lab Use Only.
RLX-33 is a selective small-molecule nonpeptide antagonist of neuropeptide relaxin-3/RXFP3 with IC50 of 2.36 uM (cAMP functional assays), selective for RXFP3 over RXFP1 and RXFP4.
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RLX-33 is a selective small-molecule nonpeptide antagonist of neuropeptide relaxin-3/RXFP3 with IC50 of 2.36 uM (cAMP functional assays), selective for RXFP3 over RXFP1 and RXFP4.
RLX-33 has favorable pharmacokinetic properties for behavioral assessment.
RLX-33 blocked food intake induced by the RXFP3-selective agonist R3/I5.
| M.Wt | 462.890 | |
| Formula | C24H19ClN4O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Elaine A. Gay, J. Med. Chem. 2022, May 20, 2022
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