RO 6842262 | LPAR1 antagonist | Probechem Biochemicals

Chemical Structure : RO 6842262

CAS No.: 1396006-71-5

RO 6842262 (RO6842262)

Catalog No.: PC-27239Not For Human Use, Lab Use Only.

RO 6842262 is a highly selective, orally active lysophosphatidic acid receptor 1 (LPAR1, LPA1) antagonist with IC50 of 25 nM, reduces plasma histamine levels in a murine LPA challenge model.

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10 mg	$398	In stock
25 mg	$598	In stock
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Biological Activity

RO 6842262 is a highly selective, orally active lysophosphatidic acid receptor 1 (LPAR1, LPA1) antagonist with IC50 of 25 nM, reduces plasma histamine levels in a murine LPA challenge model.

Physicochemical Properties

M.Wt	482.54
Formula	C28H26N4O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-1-(4'-(4-methyl-5-(((1-phenylethoxy)carbonyl)amino)-1H-1,2,3-triazol-1-yl)-[1,1'-biphenyl]-4-yl)cyclopropane-1-carboxylic acid

References

1. Yimin Qian, et al. J Med Chem. 2012 Sep 13;55(17):7920-39.

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RO 6842262 (RO6842262)

Biological Activity

Physicochemical Properties

References

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