Chemical Structure : Ralaniten acetate
Catalog No.: PC-60530Not For Human Use, Lab Use Only.
Ralaniten acetate (EPI-506) is the acetate prodrug of Ralaniten (EPI-002), a small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor for the treatment of advanced prostate cancer.
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Ralaniten acetate (EPI-506) is the acetate prodrug of Ralaniten (EPI-002), a small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor for the treatment of advanced prostate cancer.
AR NTD-targeting agents have the potential to overcome shortcomings of current hormonal therapies by inhibiting all forms of AR-mediated transcriptional activity, and as a result, may affect a broader AR population including mutational and splice variant ARs.
M.Wt | 521.003 | |
Formula | C27H33ClO8 | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
1. Antonarakis ES, et al. Oncologist. 2016 Dec;21(12):1427-1435.
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