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Ralaniten acetate

Chemical Structure : Ralaniten acetate

CAS No.: 1637573-04-6

Ralaniten acetate (EPI-506;EPI 506;EPI506)

Catalog No.: PC-60530Not For Human Use, Lab Use Only.

Ralaniten acetate (EPI-506) is the acetate prodrug of Ralaniten (EPI-002), a small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor for the treatment of advanced prostate cancer.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    Ralaniten acetate (EPI-506) is the acetate prodrug of Ralaniten (EPI-002), a small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor for the treatment of advanced prostate cancer.
    AR NTD-targeting agents have the potential to overcome shortcomings of current hormonal therapies by inhibiting all forms of AR-mediated transcriptional activity, and as a result, may affect a broader AR population including mutational and splice variant ARs.

    Physicochemical Properties

    M.Wt 521.003
    Formula C27H33ClO8
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    (R)-3-(4-(2-(4-((S)-2-acetoxy-3-chloropropoxy)phenyl)propan-2-yl)phenoxy)propane-1,2-diyl diacetate

    References

    1. Antonarakis ES, et al. Oncologist. 2016 Dec;21(12):1427-1435.

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