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Chemical Structure : SAR-100842
CAS No.: 1195941-38-8
Catalog No.: PC-35275Not For Human Use, Lab Use Only.
Fipaxalparant (SAR100842) is a potent, selective, orally available antagonist of the Lysophosphatidic Acid 1 Receptor (LPA1 receptor) with IC50 of 31 nM in β-arrestin assays.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $248 | In stock | |
| 10 mg | $398 | In stock | |
| 25 mg | $598 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
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Fipaxalparant (SAR100842) is a potent, selective, orally available antagonist of the Lysophosphatidic Acid 1 Receptor (LPA1 receptor) with IC50 of 31 nM in β-arrestin assays.
Fipaxalparant (SAR100842) demonstrates potential for the treatment of systemic sclerosis and related fibrotic diseases.
| M.Wt | 445.515 | |
| Formula | C27H27NO5 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
2-{4-methoxy-3-[2-(3-methylphenyl)ethoxy]benzamido}-2,3-dihydro-1H-indene-2-carboxylic acid |
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1. Ellery J, et al. Eur J Pharmacol. 2018 May 26;833:8-15.
2. Kihara Y, et al. Exp Cell Res. 2015 May 1;333(2):171-7.
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