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Chemical Structure : SR-2890
Catalog No.: PC-60580Not For Human Use, Lab Use Only.
SR-2890 is a potent, highly selective casein kinase 1δ/1ε (CK1δ/ε) inhibitor with IC50 of 4 nM for CK1δ.
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SR-2890 is a potent, highly selective casein kinase 1δ/1ε (CK1δ/ε) inhibitor with IC50 of 4 nM for CK1δ.
SR-2890 inhibits melanoma A375 cell growth with EC50 of 38 nM in MTT assays.
SR-2890 has physical, in vitro and in vivo PK properties suitable for use in proof of principle animal xenograft studies against human cancer cell lines.
| M.Wt | 477.932 | |
| Formula | C23H21ClFN9 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Bibian M, et al. Bioorg Med Chem Lett. 2013 Aug 1;23(15):4374-80.
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