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Susineridine

Chemical Structure : Susineridine

CAS No.: 2667632-87-1

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Susineridine (YZJ-4729, YZJ4729)

Catalog No.: PC-26358Not For Human Use, Lab Use Only.

Susineridine (YZJ-4729) is a G protein-biased μ-opioid receptor (MOR) agonist with EC50 of 17 nM, also demonstrates certain antagonistic effects on KOR and DOR, with IC50 of 1.100 μM and 6.962 μM, respectively.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    Susineridine (YZJ-4729) is a G protein-biased μ-opioid receptor (MOR) agonist with EC50 of 17 nM, also demonstrates certain antagonistic effects on KOR and DOR, with IC50 of 1.100 μM and 6.962 μM, respectively.

    Physicochemical Properties

    M.Wt 408.59
    Formula C25H36N4O
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    4H-Pyrrolo[1,2-b]pyrazol-4-amine, 5,6-dihydro-6-(1-methylethyl)-N-[2-[(9R)-9-(2-pyridinyl)-6-oxaspiro[4.5]dec-9-yl]ethyl]-, (4S,6S)-

    References

    1. Ni Y, et al. Front Pharmacol. 2024 Jan 9;14:1295319.

    2. Patent WO2023284788 A1.

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