TGR5 agonist 45h

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Chemical Structure : TGR5 agonist 45h

Catalog No.: PC-20448Not For Human Use, Lab Use Only.

TGR5 agonist 45h is a potent, selective and orally bioavailable TGR5 (GPBAR1) agonist with cAMP EC50 of 15 and 1 nM for hTGR5 and mTGR5, respectively.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

TGR5 agonist 45h is a potent, selective and orally bioavailable TGR5 (GPBAR1) agonist with cAMP EC50 of 15 and 1 nM for hTGR5 and mTGR5, respectively.

Physicochemical Properties

M.Wt	577.61
Formula	C31H30F3N5O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	trans-4-[4-[6-[(2S)-2-[[[2-(4-Cyanophenyl)ethyl]amino]carbonyl]-1-azetidinyl]-2-(trifluoromethyl)-4-pyrimidinyl]phenyl]cyclohexanecarboxylic acid

References

1. Dean P Phillips, et al. J Med Chem. 2014 Apr 24;57(8):3263-82.

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TGR5 agonist 45h

Biological Activity

Physicochemical Properties

References

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