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Chemical Structure : THIQ
Catalog No.: PC-70060Not For Human Use, Lab Use Only.
A potent and selective melanocortin 4 receptor (MC4R) agonist with EC50 of 2.1 nM.
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A potent and selective melanocortin 4 receptor (MC4R) agonist with EC50 of 2.1 nM; high selectivity over other melanocortin receptors (1184-fold vs MC3R, 350-fold vs MC5R); enhances intracavernosal pressure and stimulates erectile activity in rats ex copula.
| M.Wt | 589.181 | |
| Formula | C33H41ClN6O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Sebhat IK, et al. J Med Chem. 2002 Oct 10;45(21):4589-93.
2. Martin WJ, et al. Eur J Pharmacol. 2002 Nov 1;454(1):71-9.
3. Molden BM, et al. Mol Endocrinol. 2015 Nov;29(11):1619-33.
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