TM38837 | CB1 inverse agonist | Probechem Biochemicals

Chemical Structure : TM38837

Catalog No.: PC-22545Not For Human Use, Lab Use Only.

TM38837 is a potent, selective peripheral cannabinoid receptor 1 (CB1) inverse agonist with IC50 of 24 nM, 200-fold selective over CB2 receptor.

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Biological Activity

TM38837 is a potent, selective peripheral cannabinoid receptor 1 (CB1) inverse agonist with IC50 of 24 nM, 200-fold selective over CB2 receptor.

M.Wt	586.40
Formula	C27H20Cl2F3N7O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-(2-Chlorophenyl)-5-(4-chlorophenyl)-4-(2H-tetrazol-5-ylmethyl)-N-[(1R)-1-[4-(trifluoromethyl)phenyl]ethyl]-1H-pyrazole-3-carboxamide

1. Micale V, et al. Front Pharmacol. 2019 Mar 20;10:207.

2. Högberg T, et al. Bioorg Med Chem Lett. 2024 Jan 15;98:129572.