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Chemical Structure : Tonapofylline
CAS No.: 340021-17-2
Catalog No.: PC-60741Not For Human Use, Lab Use Only.
Tonapofylline (BG9928) is a potent, selective and orally bioavailable adenosine A1 (A1A) receptor antagonist with Ki of 7 nM.
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|---|---|---|---|
| 5 mg | $158 | In stock | |
| 10 mg | $248 | In stock | |
| 25 mg | $428 | In stock | |
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Tonapofylline (BG9928) is a potent, selective and orally bioavailable adenosine A1 (A1A) receptor antagonist with Ki of 7 nM.
Tonapofylline (BG9928) displays 915-foldselectivity over A2A receptor, 12-fold over A2B receptor.
Tonapofylline (BG9928) increases sodium excretion and cause natriuresis without causing kaliuresis or reducing renal function.
| M.Wt | 416.522 | |
| Formula | C22H32N4O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
1,3-dipropyl-8-[1-(4-propionate)-bicyclo-[2,2,2]octyl]xanthine |
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1. Auchampach JA, et al. J Pharmacol Exp Ther. 2004 Mar;308(3):846-56.
2. Kiesman WF, et al. J Med Chem. 2006 Nov 30;49(24):7119-31.
3. Greenberg B, et al. J Am Coll Cardiol. 2007 Aug 14;50(7):600-6.
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