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Chemical Structure : Zaurategrast
CAS No.: 455264-31-0
Catalog No.: PC-45954Not For Human Use, Lab Use Only.
A potent and selective, orally bioavailable α4 integrin (α4β1/VLA-4 and, to a lesser extent, α4β7 integrin) antagonist, an ester prodrug of CT-7758.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $240 | In stock | |
| 25 mg | $472 | In stock |
Bulk size, bulk discount!
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A potent and selective, orally bioavailable α4 integrin (α4β1/VLA-4 and, to a lesser extent, α4β7 integrin) antagonist, an ester prodrug of CT-7758; is developed for the treatment of multiple sclerosis.
Multiple Sclerosis
Phase 2 Discontinued
| M.Wt | 521.4057 | |
| Formula | C26H25BrN4O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
L-Phenylalanine, N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-(2,7-naphthyridin-1-ylamino)- (9CI) |
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1. Bailey, et al. Current Immunology Reviews, 2012, 8, 135-140
2. Wolf C, et al. PLoS One. 2013;8(3):e58438.
3. Chanteux H, et al. Drug Metab Dispos. 2014 Jan;42(1):153-61.
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