β-catenin-BCL9 inhibitor 28

Chemical Structure : β-catenin-BCL9 inhibitor 28

Catalog No.: PC-28110Not For Human Use, Lab Use Only.

β-catenin-BCL9 inhibitor 28 is a potent and selective inhibitor of β-catenin/BCL9 interaction, shows high-affinity binding to β-catenin with SPR Kd of 82 nM, enhances antigen presentation and activates cDC1 cells.

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Biological Activity

β-catenin-BCL9 inhibitor 28 is a potent and selective inhibitor of β-catenin/BCL9 interaction, shows high-affinity binding to β-catenin with SPR Kd of 82 nM, enhances antigen presentation and activates cDC1 cells.

Physicochemical Properties

M.Wt	670.86
Formula	C37H50N8O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	2-(3-((R)-3-(3-(4-(1H-pyrazol-4-yl)benzyl)-3-cyclopropylureido)piperidin-1-yl)phenoxy)-N-(2-(2-(2-aminoethyl)pyrrolidin-1-yl)-2-oxoethyl)-2-methylpropanamide

References

1. Wenhua Zhu, et al. J Med Chem. 2024 Aug 8;67(15):12485-12520.

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