Cat. No. |
Product Name |
Information |
PC-24448 |
DDR1-IN-2
DDR1 inhibitor
|
DDR1-IN-2 is a potent and selective inhibitor of DDR1 receptor tyrosine kinase with IC50 of 47.6 nM, 4-fold selective over DDR-2 (IC50=145 nM), inhibits DDR1 autophosphorylation in cells. |
PC-24447 |
DDR1-IN-1
DDR1 inhibitor
|
DDR1-IN-1 is a potent and selective inhibitor of DDR1 receptor tyrosine kinase with IC50 of 105 nM, 4-fold selective over DDR-2 (IC50=413 nM), inhibits DDR1 autophosphorylation in cells. |
PC-23135 |
CH6824025
DDR1 inhibitor
|
CH6824025 is a potent, selective discoidin domain receptor 1 (DDR1) inhibitor, dose-dependently inhibits the phosphorylation of DDR1 induced by adding Type 1 collagen to U2OS cells stably expressing DDR1 with IC50 of 8.9 nM. |
PC-63520 |
LCB 03-0110 dihydrochloride
|
LCB 03-0110 is a potent, ATP-competitive inhibitor of Discoidin domain receptor (DDR) family and c-Src tyrosine kinase family, as well as Btk and Syk. |