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(1S,2S)-2-PCCA

Chemical Structure : (1S,2S)-2-PCCA

CAS No.: 1609624-97-6

(1S,2S)-2-PCCA

Catalog No.: PC-61116Not For Human Use, Lab Use Only.

The (1R,2R) diastereomer of 2-PCCA, a potent, selective agonist of the orphan GPR88 receptor with EC50 of 373 nM, 5-fold more potent than the (1S, 2S)-isomer..

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

The (1R,2R) diastereomer of 2-PCCA, a potent, selective agonist of the orphan GPR88 receptor with EC50 of 373 nM, 5-fold more potent than the (1S, 2S)-isomer.

Physicochemical Properties

M.Wt 455.646
Formula C30H37N3O
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

(1S,2S)-N-((2S,3S)-2-amino-3-methylpentyl)-N-(4'-propyl-[1,1'-biphenyl]-4-yl)-2-(pyridin-2-yl)cyclopropane-1-carboxamide

References

1. Jin C, et al. ACS Chem Neurosci. 2014 Jul 16;5(7):576-87.

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