You are here:Home-Chemical Inhibitors & Agonists-GPCR-Chemokine Receptor (CCR and CXCR)

Request The Product List ofChemokine Receptor (CCR and CXCR) Chemokine Receptor (CCR and CXCR)

Cat. No. Product Name CAS No. Information
PC-73030

CCR4-IN-31

2206788-99-8 CCR4-IN-31 (CCR4-351) is a potent, selective, orally bioavailable CCR4 antagonist with IC50 of 40 nM (Ca2+ flux).
PC-72896

CCR2 inhibitor SD-24

1237502-86-1 CCR2 inhibitor SD-24 is a potent selective CCR2 antagonist with pKi of 8.5.
PC-35600

LIT-927

2172879-52-4 LIT-927 (LIT927) is the first selective, locally and orally active CXCL12 neutraligand with Ki of 267 nM for CXCL12-TR binding inhibition.
PC-35572

CCR6 inhibitor 35

2437547-04-9 CCR6 inhibitor 35 is a potent and selective CCR6 inhibitor with IC50 of 6.0 nM (hCCR6).
PC-35514

AZ084

929300-19-6 AZ084 (AZ-084) is a potent, selective, allosteric, orally available CCR8 antagonist with Ki of 0.9 nM.
PC-35358

BL5923

868408-20-2 BL5923 (BL-5923) is a potent, highly specific, orally available inhibitor of CCR1 with IC50 of 20.4 and 22.8 nM for human and mouse CCR1, resepctively.
PC-63440

R243

688352-84-3 R243 is a potent, small molecule CCR8 antagonist that inhibits CCR8 signaling and chemotaxis, inhibits CCL1-induced Ca2+ flux and CCL1-driven peritoneal macrophages aggregation at 0.2 uM.

Request The Product List

* Indicates a Required FieldYour information is safe with us.

  • *Product List:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Country:
  • Additional Information:

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com