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Chemical Structure : ARUK2001607
Catalog No.: PC-49589Not For Human Use, Lab Use Only.
ARUK2001607 is a potent, selective and brain penetrant PI5P4Kγ inhibitor with binding KD of 7.1 nM, pIC50 of 7.1 (PI5P4Kγ+).
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ARUK2001607 is a potent, selective and brain penetrant PI5P4Kγ inhibitor with binding KD of 7.1 nM, pIC50 of 7.1 (PI5P4Kγ+).
ARUK2001607 showed excellent selectivity data against >150 kinases and a Cerep safety panel, also showed good potencies at PI5P4Kγ (WT and γ+), were selective vs PI5P4Kα and β.
| M.Wt | 319.40 | |
| Formula | C14H13N3O2S2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Timothy P C Rooney, et al. J Med Chem. 2022 Dec 14. doi: 10.1021/acs.jmedchem.2c01693.
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