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Azilsartan

Chemical Structure : Azilsartan

CAS No.: 147403-03-0

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Azilsartan (TAK-536, TAK536)

Catalog No.: PC-44124Not For Human Use, Lab Use Only.

Azilsartan (TAK-536) is a specific and potent angiotensin II type 1 receptor (AT1) antagonist with IC50 of 2.6 nM, used in the treatment of adults with essential hypertension.

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50 mg $198 In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Azilsartan (TAK-536) is a specific and potent angiotensin II type 1 receptor (AT1) antagonist with IC50 of 2.6 nM, used in the treatment of adults with essential hypertension.

Physicochemical Properties

M.Wt 456.4501
Formula C25H20N4O5
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

1H-Benzimidazole-7-carboxylic acid, 1-[[2'-(2,5-dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-

References

1. French C, et al. J Cardiovasc Pharmacol. 2011 Aug;58(2):143-8.

2. Kusumoto K, et al. Eur J Pharmacol. 2011 Nov 1;669(1-3):84-93.

3. Bönner G, et al. J Hum Hypertens. 2013 Aug;27(8):479-86.

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