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Chemical Structure : BAY-6035
Catalog No.: PC-63250Not For Human Use, Lab Use Only.
BAY-6035 is a potent, peptide-competitive inhibitor of histone methyltransferase SMYD3, inhibits in vitro methylation of MEKK2 peptide with IC50 of 88 nM, >100-fold selectivity over other HMTases.
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BAY-6035 is a potent, peptide-competitive inhibitor of histone methyltransferase SMYD3, inhibits in vitro methylation of MEKK2 peptide with IC50 of 88 nM, >100-fold selectivity over other HMTases; inhibits the methylation of MEKK2 in cells with IC50 of 70 nM.
| M.Wt | 396.491 | |
| Formula | C22H28N4O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1, Stefan Gradl, et al. SLAS Discov. 2021 Sep;26(8):947-960.
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