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BAY-876

Chemical Structure : BAY-876

CAS No.: 1799753-84-6

BAY-876 (BAY876)

Catalog No.: PC-42031Not For Human Use, Lab Use Only.

BAY-876 (BAY876) is a potent, highly selective and oral bioavailable GLUT1 inhibitor with IC50 of 2 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

BAY-876 (BAY876) is a  potent, highly selective and oral bioavailable GLUT1 inhibitor with IC50 of 2 nM.
BAY-876 displays >100-fold selectivity against GLUT2, GLUT3, and GLUT4.
BAY-876 exhibits good metabolic stability in vitro and high oral bioavailability in vivo.

Physicochemical Properties

M.Wt 496.4164
Formula C24H16F4N6O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

DMSO: ≥ 100 mg/mL

Chemical Name/SMILES

2,4-Quinolinedicarboxamide, N4-[1-[(4-cyanophenyl)methyl]-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl]-7-fluoro-

References

1. Siebeneicher H, et al. ChemMedChem. 2016 Oct 19;11(20):2261-2271.

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