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Cat. No. Product Name CAS No. Information
PC-35327

WZB117

1223397-11-2 WZB117 (WZB-117) is a small-molecule inhibitor of glucose transporter 1 (GLUT1), inhibits glucose transport and cancer cell proliferation with IC50 of 10 uM; decreases in levels of Glut1 protein, intracellular ATP, and glycolytic enzymes in treated cancer cells, inhibits cancer growth in tumor-bearing nude mice; also inhibits the self-renewal and tumor-initiating capacity of cancer stem cells (CSCs).
PC-62895

Fasentin

392721-37-8 Fasentin is a novel inhibitor of glucose uptake (GLUT) that sensitizes cancer cells to FAS-induced cell death, preferentially inhibits GLUT4 (IC50=68 uM) over GLUT1; sensitizes cancer cells to the death ligands FAS and TNF apoptosis-inducing ligand, and induces G1 cell cycle arrest.
PC-60884

GLUT4-IN-17

1061081-61-5 A potent, selective glucose transporter 4 (GLUT4) inhibitor with IC450 of 10.8 uM, inhibits MM cell proliferation; reduces ATB-BMPA binding to GLUT4 to a much greater extent than to GLUT1, inhibits 2-DOG uptake in GLUT4-expressing cells.
PC-45543

STF-31

724741-75-7 A selective GLUT1 inhibitor that does not bind to other glucose transporters; selectively kills RCCs by specifically targeting glucose uptake through GLUT1 and exploiting the unique dependence of these cells on GLUT1 for survival; also inhibits the enzymatic activity of NAMPT in a biochemical assay in vitro.
PC-42031

BAY-876

1799753-84-6 A potent, highly selective and oral bioavailable GLUT1 inhibitor with IC50 of 2 nM; displays >100-fold selectivity against GLUT2, GLUT3, and GLUT4; exhibits good metabolic stability in vitro and high oral bioavailability in vivo.

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