Chemical Structure : BCAT2-IN-1
CAS No.:
1875078-61-7
BCAT2-IN-1
(BCATm inhibitor)
Catalog No. : PC-26618Not For Human Use, Lab Use Only.
BCAT2-IN-1 is a potent, selective, in-vivo efficacious BCATm (BCAT2) inhibitor with pIC50 of 7.3, 100-fold selective for BCATm over BCATc.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-2661801
Biological Activity
BCAT2-IN-1 is a potent, selective, in-vivo efficacious BCATm (BCAT2) inhibitor with pIC50 of 7.3, 100-fold selective for BCATm over BCATc.
Physicochemical Properties
M.Wt
538.46
Formula
C25H24BrN5O2S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
1H-Benzimidazole-5-carboxamide, 1-[(1R,3S)-3-[[(5-bromo-2-thienyl)carbonyl]amino]cyclohexyl]-N-methyl-2-(2-pyridinyl)-, rel-
References
1. Hongfeng Deng, et al. ACS Med Chem Lett. 2016 Feb 8;7(4):379-84.
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