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Chemical Structure : BRD9-IN-28
Catalog No.: PC-62938Not For Human Use, Lab Use Only.
BRD9-IN-28 is a highly potent and selective BRD7/9 bromodomain inhibitor with pIC50 of 6.9, Kd of 68 nM for BRD9.
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BRD9-IN-28 is a highly potent and selective BRD7/9 bromodomain inhibitor with pIC50 of 6.9, Kd of 68 nM for BRD9.
BRD9-IN-28 is slightly less potent against BRD7 (Kd=368 nM) and completely inactive against BAZ2B, little affinity across BRD proteins from sub-families 1-3 and 5-8, including BAZ2A and BAZ2B.
BRD9-IN-28 shows weak affinity for the BRDs from CBP, p300 and FALZ.
| M.Wt | 360.417 | |
| Formula | C21H20N4O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Duncan. A. Hay, et al. Med. Chem. Commun., 2015, DOI: 10.1039/C5MD00152H.
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