Welcome to Shanghai Probechem Biochemicals Co Ltd !Global Supplier of Chemical Probes, Inhibitors & Agonists.
Chemical Structure : BRD9539
CAS No.: 1374601-41-8
Catalog No.: PC-49729Not For Human Use, Lab Use Only.
BRD9539 is a small molecule inhibitor of histone hethyltransferase of G9a (euchromatin histone methyltransferase 2, EHMT2) with IC50 of 6.3 uM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 25 mg | $258 | In stock | |
| 50 mg | $428 | In stock | |
| 100 mg | $728 | In stock | |
| 250 mg | Get quote | ||
| 1 g | Get quote |
Bulk size, bulk discount!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
BRD9539 is a small molecule inhibitor of histone hethyltransferase of G9a (euchromatin histone methyltransferase 2, EHMT2) with IC50 of 6.3 uM.
BRD9539 also inhibits PRC2 activity with a similar IC50, displays no inhibition aginst SUV39H1 and DNMT1.
BRD9539 is a more potent biochemical inhibitor than its methyl-ester analogue BRD4770.
| M.Wt | 399.45 | |
| Formula | C24H21N3O3 | |
| Appearance | Solid | |
| Storage |
|
|
| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
2-benzamido-1-(3-phenylpropyl)-1H-benzo[d]imidazole-5-carboxylic acid |
|
1. Yuan Yuan, et al. ACS Chem Biol. 2012 Jul 20;7(7):1152-7.
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright
