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Chemical Structure : Bitopertin R enantiomer
Catalog No.: PC-42707Not For Human Use, Lab Use Only.
A potent and selective GlyT1 inhibitor with EC50 of 54 nM.
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A potent and selective GlyT1 inhibitor with EC50 of 54 nM; no activity for GlyT2, hERG, CYP450 enzymes above 10 uM; the R enantiomer of RG-1678.
Schizophrenia
Phase 3 Clinical
| M.Wt | 543.455 | |
| Formula | C21H20F7N3O4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Pinard E, et al. J Med Chem. 2010 Jun 24;53(12):4603-14.
2. Alberati D, et al. Neuropharmacology. 2012 Feb;62(2):1152-61
3. Martin-Facklam M, et al. Neuropsychopharmacology. 2013 Feb;38(3):504-12.
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