You are here:Home-ADCs and PROTACs-E3 Ligase Ligand-DCAF1 ligand 1
DCAF1 ligand 1

Chemical Structure : DCAF1 ligand 1

CAS No.:

DCAF1 ligand 1 (DCAF1 E3 ligase binder 1)

Catalog No.: PC-21643Not For Human Use, Lab Use Only.

DCAF1 ligand 1 is a selective DCAF1 E3 ligase receptor binder with SPR KD value of 0.03 uM.

Packing Price Stock Quantity
50 mg Get quote
100 mg Get quote
200 mg Get quote
1 g Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC)

Biological Activity

DCAF1 ligand 1 is a selective DCAF1 E3 ligase receptor binder with SPR KD value of 0.03 uM.
DCAF1 E3 ligase binder 1 shows only partial overlap with recently reported DCAF1 ligand OICR-8268 (Cat# PC-20292).
DCAF1 E3 ligase binder 1 displays no activity against any other WDR-containing proteins.

Physicochemical Properties

M.Wt 507.08
Formula C28H35ClN6O
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

1-(4-(4-((2-aminoethyl)amino)-2-(1-(4-chlorophenyl)cyclohexyl)quinazolin-7-yl)piperazin-1-yl)ethan-1-one

References

1. Schröder M, et al. Nat Commun. 2024 Jan 4;15(1):275.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: